Department of Pharmaceutical Chemistry - Pharmacy

Cairo, Abbassia, EG

OrgUnit's Researchers publications
(Dept/Workgroup Publication)

Results 121-140 of 191 (Search time: 0.0 seconds).

Issue DateTitleAuthor(s)
121Oct-2022New fluorinated diarylureas linked to pyrrolo[2,3-d]pyrimidine scaffold as VEGFR-2 inhibitors: Molecular docking and biological evaluationAdel, Mai; Abouzid, Khaled 
122Dec-2007A NEW SCAFFOLD FOR D3 DOPAMINERGIC AFFINITY CONTAINING ARYLPIPERAZINE FRAGMENT: MOLECULAR MODELING, SYNTHESIS, IN VITRO AND IN VIVO PHARMACOLOGICAL EVALUATIONAbou El Ella, Dalal ; Franziska K. U. Müller
123Dec-2022Novel 1,3-diaryl pyrazole derivatives bearing methylsulfonyl moiety: Design, synthesis, molecular docking and dynamics, with dual activities as anti-inflammatory and anticancer agents through selectively targeting COX-2Shaker, Ahmed M M; Shahin, Mai I. ; AboulMagd, Asmaa M; Abdel Aleem, Seham A; Abdel-Rahman, Hamdy M; Abou El Ella, Dalal 
1242013Novel 2-thiopyrimidine derivatives as CDK2 inhibitors: molecular modeling, synthesis, and anti-tumor activity evaluationFathalla, OAM; Ismail, MAH; Anwar, MM; Abouzid, Khaled ; Ramadan, AAK
12515-May-2008Novel anti-inflammatory agents based on pyridazinone scaffold; design, synthesis and in vivo activityAbouzid, Khaled ; Bekhit, Salma A
1262020Novel Benzimidazole/Hydrazone Derivatives as Promising Anticancer Lead Compounds: Design, Synthesis, and Molecular Docking StudyMorcoss, Martha; Abdelhafez, El Shimaa; Abdel-Rahman, Hamdy; lhab Abdel Aziz Mohammed ; Abou El Ella, Dalal 
1271-Feb-2024Novel indolinone-tethered benzothiophenes as anti-tubercular agents against MDR/XDR M. tuberculosis: Design, synthesis, biological evaluation and in vivo pharmacokinetic studyEldehna, Wagdy M.; Mahmoud, Sally Tarek; Elshnawey, Esraa R.; Elsayed, Zainab M.; Majrashi, Taghreed A.; El-Ashrey, Mohamed K.; Rashed, Mahmoud; Hemeda, Loah R.; Shoun, Aly A.; Elkaeed, Eslam B.; El Hassab, Mahmoud A.; Abdel-Aziz, Marwa M.; Shahin, Mai I. 
1281-Dec-2017Novel quinoline-3-carboxamides (Part 2): Design, optimization and synthesis of quinoline based scaffold as EGFR inhibitors with potent anticancer activityAly, Rasha M.; Serya, Rabah ; El-Motwally, Amira M.; Abbas, Safinaz; Abou El Ella, Dalal ; Esmat, Ahmed 
12915-Jul-2018Novel series of 6-(2-substitutedacetamido)-4-anilinoquinazolines as EGFR-ERK signal transduction inhibitors in MCF-7 breast cancer cellsIsmail, Rania S M; Abou-Seri, Sahar M; Eldehna, Wagdy M; Ismail, Nasser S M; Elgazwi, Sara M; Ghabbour, Hazem A; Ahmed, Mahmoud Salama; Halaweish, Fathi T; Abou El Ella, Dalal 
13015-Mar-2024Novel sulfonamide-indolinone hybrids targeting mitochondrial respiration of breast cancer cellsHelmy, Sama W.A.; Abdel-Aziz, Amal Kamal ; Dokla, Eman M.E.; Ahmed, Tarek E.; Hatem, Yasmin; Abdel Rahman, Engy A.; Sharaky, Marwa; Shahin, Mai I. ; Elrazaz, Eman Z.; Serya, Rabah A.T.; Henary, Maged; Ali, Sameh S.; Abou El Ella, Dalal A.
1312011Optimization of Benzoisothiazole dioxide inhibitory activity of the NS5B polymerase of HCV genotype 4 using ligand-steered homological modeling, reaction-driven scaffold-hopping and Enovo workflowMahmoud, Amr Hamed; Abouzid, Khaled ; El Ella, Dalal Abd El Rahman Abou; Hamid Ismail, Mohamed Abdel
1322010Organic synthesis and biological evaluation of novel "3+1" mixed ligands of technetium-99m Gabapentin as receptor imaging agentsAmin, AM; Abouzid, Khaled ; Bayoumi, NA; Abd El-hamid, M
1331-Aug-2020Penicillin binding protein 2a: An overview and a medicinal chemistry perspectiveShalaby, Menna-Allah W; Dokla, Eman ; Serya, Rabah ; Khaled A M Abouzid 
1341-Dec-2019Phosphatidylinositol 3 kinase (PI3K) inhibitors as new weapon to combat cancerElmenier, Fatma M; Lasheen, Deena S. ; Khaled A M Abouzid 
1351-Sep-2011Preparation of 99mTc-ceftazidime as a model of infection imaging agentM. A. Motaleb; A. A. El Mohty; M. A. El Garhy; Mohamed abdel Hamid Ismail; Abouzid, Khaled ; Tamer M. Sakr
162016Pyrazolo[3,4-d]pyrimidine based scaffold derivatives targeting kinases as anticancer agentsIsmail, Nasser S.M.; Ali, Eslam M.H.; Ibrahim, Diaa A.; Serya, Rabah A.T.; Abou El Ella, Dalal 
17Mar-2017Pyridazine Based Scaffolds as Privileged Structures in anti-Cancer TherapyJaballah, Maiy Youssef; Serya, Rabah Taha; Abouzid, Khaled 
181-Jan-2008Pyridazinone derivatives: design, synthesis, and in vitro vasorelaxant activityAbouzid, Khaled ; Abdel Hakeem, Maha; Khalil, Omnya; Maklad, Yosria
1916-Aug-2024Pyridazinone-based derivatives as anticancer agents endowed with anti-microbial activity: molecular design, synthesis, and biological investigationEl-Nagar, Mohamed K.S.; Shahin, Mai I. ; El-Behairy, Mohammed F.; Taher, Ehab S.; El-Badawy, Mohamed F.; Sharaky, Marwa; Abou El Ella, Dalal A.; Abouzid, Khaled A.M.; Adel, Mai
20Sep-2018Pyrrolopyrimidine, A Multifaceted Scaffold in Cancer Targeted TherapyAdel, Mai; Serya, Rabah A T; Lasheen, Deena S. ; Abouzid, Khaled