Issue Date Title Author(s) 1 31-Dec-2026 Multi-targeted pyrazole scaffolds: synthesis, mechanistic insights, and therapeutic potential in anticancer, antioxidant, and anti-inflammatory applications Aljameel, Suhailah S; Eissa, Mohamed E; Alatawi, Zinab; Alahmadi, Hanadi A; Azab, Mohammad E ; Yousef, Tarek A; Aljohi, Hasan A; Al-Farraj, Eida S; Bahattab, Eman Abdullah; Ghareeb, Ahmed; El-Helw, Eman A. E. ; Sayed Karam Ramadan Emam ; Eman A. E. El-Helw
2 24-Apr-2026 Exploring insecticidal activity and SAR study of newly synthesized Benzo[h]quinoline-based heterocycles against Aphis craccivora Koch. and Culex pipiens L. Larvae Abdel-Haleem, Doaa R; Khalil, A. K. ; Sayed Karam Ramadan Emam ; Eman A. E. El-Helw
3 2026 Green Synthesis and Biological Assessment of Curcumin-Based Heterocycles via a Microwave-Ultrasonic-Ultraviolet Reactor: DFT, Docking, and MD Insights Saleh, Esraa M.; Fahim, Asmaa M.; Awady, Mohamed E. El; El-Banna, Mohamed G.; Rizk, Sameh Ahmed ; Eman A. E. El-Helw
4 2026 Multitarget bioactive benzo [f] quinoline heterocycles from a thiocarbohydrazone scaffold: synthesis, biological assays, and in silico mechanistic rationale Saleh, Esraa M; El-Banna, Mohamed G; Fahim, Asmaa M; El Awady, Mohamed E; Rizk, Sameh A; Eman A. E. El-Helw
5 2026 Synthesis and biological evaluation of novel heterocyclic compounds derived from ammonium thiocyanate for control of Culex pipiens and Musca domestica. Ghareeb, Eman A; Kamal, Mahmoud; Farag, Shaimaa M; Ammar, Asmaa M; Mahmoud, Naglaa FH; Eman A. E. El-Helw
6 2026 Synthesis and In Silico Studies of New Tetrahydrobenzo[ b ]Thiophenes and Heteroannulated Candidates as Antiproliferative Agents Elgubbi, Amna S.; Gomha, Sobhi M.; Zaki, Magdi E. A.; Sayed Karam Ramadan Emam ; Eman A. E. El-Helw
7 29-Nov-2025 Synthesis and insecticidal activity of some pyrazole, pyridine, and pyrimidine candidates against Culex pipiens L. larvae Eman A. E. El-Helw ; El-Bordany, Eman A; El-Fagal, Sara F; Ghareeb, Eman A; Doaa Ramadan Abdel Haleem Ramadan
8 24-Nov-2025 Synthesis, antiproliferative screening, and molecular docking of some heterocycles derived from N-(1-(5-chloro-3-methyl-1-phenyl-1H-pyrazol-4-yl)-3-hydrazineyl-3-oxoprop-1-en-2-yl)benzamide Eman A.E. El-Helw ; Youssef, Youssef M; Elsayed, Galal A. ; El-Sayed, Amira A; Hassaballah, Aya I; Mohamed, Ashraf M; Azab, Mohammad E
9 Nov-2025 Multi-Target Rational Design and Synthesis of Some 2-Quinolinone Antitumor Candidates Downregulating the Expression of EGFR, VEGFR-2, and Telomerase With Apoptotic Potential Eman A.E. El-Helw ; Mousa, Mai H A; Ghareeb, Eman A; Mahmoud, Naglaa F H; Sharaky, Marwa; El-Bordany, Eman A; Khatib, Arwa Omar Al; Soliman, Elsayed A; Alnajjar, Radwan; Al-Karmalawy, Ahmed A
10 Oct-2025 Straightforward synthesis and in silico evaluation of pyrazolylthiazolidinone derivatives as prospective antiproliferative agents Ramadan, Sayed K. ; Gomha, Sobhi M; Eman A. E. El-Helw
11 29-Sep-2025 Straightforward synthesis and in silico evaluation of pyrazolylthiazolidinone derivatives as prospective antiproliferative agents Ramadan, Sayed ; Gomha, Sobhi M; El-Helw, Eman A. E.
12 13-May-2025 Antioxidant activity, molecular docking, and modeling pharmacokinetics study of some benzo[f]quinoline candidates El-Fagal, Sara F; Eman A. E. El-Helw ; El-Bordany, Eman A; Ghareeb, Eman A
13 24-Mar-2025 Synthesis of Benzo[h]quinoline derivatives and evaluation of their insecticidal activity against Culex pipiens L. larvae Hosni, Eslam M; E.A.E. El-Helw ; Ramadan, Sayed ; Hashem, Ahmed ; Wael Abou-Elmagd
14 1-Jan-2025 Synthesis and In Silico Evaluation of Thiazole, Thiazolidinone, and Pyrimidinethione Candidates Bearing A Benzo[h]Quinoline Scaffold as Potential Antiproliferative Agents Gomha, Sobhi M.; Ali, Amira T.; Sayed Karam Ramadan Emam ; Eman A. E. El-Helw
15 2025 In Silico ADME, DFT, and Antiproliferative Activity of Pyrazole-based Pyrimidinethione, Triazolethione, and Thiadiazolopyrimidine Derivatives Ramadan, Sayed ; Gomha, S. M.; E.A.E. El-Helw
16 2025 Synthesis and Exploring Antiproliferative Activity of Some Pyrazole-Bearing Heterocycles: DFT, Molecular Docking, and ADME Study Ramadan, Sayed ; Gomha, S. M.; El-Helw, E.A.E.
17 2025 Design, Synthesis, Antiproliferative Activity and In Silico Studies of 2-Oxo-1,2-Dihydroquinolin Derivatives Eman A. E. El-Helw ; Ghareeb, Eman A.; Mahmoud, Naglaa F. H.; El-Bordany, Eman A.; Soliman, Elsayed A.; El-Khouly, Ahmed; Abouzid, Khaled
18 2025 Design, synthesis, and in silico studies of pyrazolyl-thiazole and thiazolidinone hybrids as potential antiproliferative agents Ramadan, Sayed K; Ali, Amira T; Gomha, Sobhi M; Ramadan, S.K. ; Eman A. E. El-Helw
19 5-Jul-2024 Synthesis and in silico studies of certain benzo[f]quinoline-based heterocycles as antitumor agents Asran, Mahmoud; Helal, Maher H; Alzahrani, Abdullah Y A; Ramadan, Sayed ; Azab, Mohammad ; Eman A. E. El-Helw
20 6-Jun-2024 β-Enaminonitrile in the synthesis of tetrahydrobenzo[b]thiophene candidates with DFT simulation, in vitro antiproliferative assessment, molecular docking, and modeling pharmacokinetics Elgubbi, Amna S.; Abousiksaka, Motaleb S.; Alzahrani, Abdullah Y. A.; Sayed Karam Ramadan Emam ; Eman A. E. El-Helw