Issue Date Title Author(s) 21 2022 3-Aryl/hetaryl-2-cyanoacryloyl chlorides: Synthesis and Reactions with Binucleophiles Targeting Heterocycles El-Ziaty, Ahmed ; S.K. Ramadan ; Eman A.E. El-Helw
22 2022 Facile Synthesis, Biological Evaluation, DFT Studies and in Silico Prediction ADME/Pharmacokinetics Properties of N-(1-(2-Chlorobenzo[h]Quinolin-3-yl)-1-Substituted-vin-2-yl)Benzamide Derivatives Abdelrahman, AM; Fahmi, AA; Rizk, Sameh Ahmed ; Eman A. E. El-Helw
23 2022 Synthesis and Antiproliferative Screening of Some Heterocycles Derived from 4-((5-Chloro-3-Methyl-1-Phenyl-1H-Pyrazol-4-yl)Methylene)-2-Phenyloxazol-5(4H)-One Youssef, YM; Azab, ME; Elsayed, GA; El-Sayed, AA; Eman A. E. El-Helw
24 2023 Synthesis, Cytotoxic, and Antioxidant Activity of Some Benzoquinoline-Based Heterocycles Asran, Mahmoud; Azab, Mohammad E.; Helal, Maher H.; Sayed K. Ramadan ; Eman A. E. El-Helw
25 1-Jan-2023 Synthesis and antioxidant activity of some pyrazole-based heterocycles using a 2(3H)-furanone building block Youssef, Youssef M.; Elsayed, Galal A. ; El-Sayed, Amira A.; Hassaballah, Aya I.; Azab, Mohammad ; Eman A. E. El-Helw
26 1-Jan-2023 Synthesis, Density Functional Theory, Insecticidal Activity, and Molecular Docking of Some N-Heterocycles Derived from 2-((1,3-Diphenyl-1H-Pyrazol-4-yl)Methylene)Malonyl Diisothiocyanate Abdelrahman, Aya M.; Fahmi, Abdelgawad A.; Rizk, Sameh Ahmed ; Eman A. E. El-Helw
27 1-Jan-2023 Synthesis, DFT and Antitumor Activity Screening of Some New Heterocycles Derived from 2,2'-(2-(1,3-Diphenyl-1H-Pyrazol-4-yl)Ethene-1,1-Diyl)Bis(4H-Benzo[d][1,3]Oxazin-4-One) Abdelrahman, Aya M.; Fahmi, Abdelgawad A.; Rizk, Sameh Ahmed ; Eman A. E. El-Helw
28 1-Sep-2023 Synthesis and antioxidant, antimicrobial, and antiviral activity of some pyrazole-based heterocycles using a 2(3H)-furanone derivative Youssef, Youssef M.; Azab, Mohammad E.; Elsayed, Galal A. ; El-Sayed, Amira A.; Hassaballah, Aya I.; El-Safty, Mounir M.; Soliman, Reem A.; El-Helw, EAE
29 12-Sep-2023 Synthesis and cytotoxicity evaluation of novel 1,8-acridinedione derivatives bearing phthalimide moiety as potential antitumor agents Khatab, Hassan A; Hammad, Sherif F; El-Fakharany, Esmail M; Hashem, Ahmed I. ; El-Helw, EAE
30 2024 Synthesis, insecticidal Activity, and molecular docking analysis of some benzo[h]quinoline derivatives against Culex pipiens L. Larvae Hosni, Eslam M.; Mahmoud Kamal ; Hashem, Ahmed I. ; Sayed Karam Ramadan Emam ; Eman A.E. El-Helw
31 1-Jan-2024 Some Thiazolopyrimidine Derivatives: Synthesis, DFT, Cytotoxicity, and Pharmacokinetics Modeling Study Ramadan, Sayed ; Alzahrani, Abdullah Y. A.; Eman A. E. El-Helw
32 1-Jan-2024 Synthesis, antiproliferative activity, and in silico studies of quinoline-based pyrimidinedione and thiazolidinedione derivatives Alzahrani, Abdullah Y.A.; Ramadan, S.K. ; Eman A. E. El-Helw
33 1-Jan-2024 Synthesis and Biological Applications of Coumarinyl-Chalcones Ramadan, Sayed ; Rizk, Sameh Ahmed ; Eman A. E. El-Helw
34 1-Jan-2024 Facile Synthesis and Antioxidant Activity Screening of Some Novel 3-Substituted Indole Derivatives Elgubbi, Amna S.; Alzahrani, Abdullah Y.A.; Eman A. E. El-Helw ; Shaban, Safaa S.
35 14-Feb-2024 Synthesis, computational chemical study, antiproliferative activity screening, and molecular docking of some thiophene-based oxadiazole, triazole, and thiazolidinone derivatives Elgubbi, Amna S; Alzahrani, Abdullah Y A; Ramadan, Sayed ; Eman A.E. El-Helw
36 6-Jun-2024 β-Enaminonitrile in the synthesis of tetrahydrobenzo[b]thiophene candidates with DFT simulation, in vitro antiproliferative assessment, molecular docking, and modeling pharmacokinetics Elgubbi, Amna S.; Abousiksaka, Motaleb S.; Alzahrani, Abdullah Y. A.; Sayed Karam Ramadan Emam ; Eman A. E. El-Helw
37 2025 In Silico ADME, DFT, and Antiproliferative Activity of Pyrazole-based Pyrimidinethione, Triazolethione, and Thiadiazolopyrimidine Derivatives Ramadan, Sayed ; Gomha, S. M.; E.A.E. El-Helw
18 2025 Synthesis and Exploring Antiproliferative Activity of Some Pyrazole-Bearing Heterocycles: DFT, Molecular Docking, and ADME Study Ramadan, Sayed ; Gomha, S. M.; El-Helw, E.A.E.
19 2025 Design, Synthesis, Antiproliferative Activity and In Silico Studies of 2-Oxo-1,2-Dihydroquinolin Derivatives Eman A. E. El-Helw ; Ghareeb, Eman A.; Mahmoud, Naglaa F. H.; El-Bordany, Eman A.; Soliman, Elsayed A.; El-Khouly, Ahmed; Abouzid, Khaled
20 Jan-2025 Synthesis, in vivo evaluation, and in silico molecular docking of benzo[h]quinoline derivatives as potential Culex pipiens L. larvicides Hosni, Eslam M; E.A.E. El-Helw ; Ramadan, Sayed K.; Abou-Elmagd, Wael S. I.; Hashem, Ahmed I.