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| | Issue Date | Title | Author(s) |
| 21 | 1-Dec-2021 | Indolin-2-one derivatives as selective Aurora B kinase inhibitors targeting breast cancer | Dokla, Eman ; Abdel-Aziz, Amal Kamal ; Milik, Sandra N.; Mahmoud, Amr H.; Saadeldin, Mona Kamal; McPhillie, Martin J.; Minucci, Saverio; Khaled A M Abouzid |
| 22 | Jun-2014 | Molecular design and synthesis of 1,4-disubstituted piperazines as α(1)-adrenergic receptor blockers | Hussein, Mohammed M; Serya, Rabah ; Abdel Naby, Rana M; Al-Abd, Ahmed M; Saleh, Dalia O; El-Eraky, Wafaa I; Khaled A M Abouzid ; Abou El Ella, Dalal |
| 23 | 2026 | Multitarget bioactive benzo [f] quinoline heterocycles from a thiocarbohydrazone scaffold: synthesis, biological assays, and in silico mechanistic rationale | Saleh, Esraa M; El-Banna, Mohamed G; Fahim, Asmaa M; El Awady, Mohamed E; Rizk, Sameh A; Eman A. E. El-Helw |
| 24 | 16-Jul-2021 | New N-(1,3,4-thiadiazol-2-yl)furan-2-carboxamide derivatives as potential inhibitors of the VEGFR-2 | Soliman Farag Saad, Paula ; Hemdan, Magdy M. ; El-Sayed, Wael ; Mohamed Hussein Hussein Moustafa Hekal |
| 25 | Apr-2023 | New trends in synthetic drugs and natural products targeting 20S proteasomes in cancers | Atta, Hind; Alzahaby, Nouran ; Hamdy, Nadia M; Emam, Soha H; Sonousi, Amr; Ziko, Laila |
| 6 | Dec-2022 | Novel 1,3-diaryl pyrazole derivatives bearing methylsulfonyl moiety: Design, synthesis, molecular docking and dynamics, with dual activities as anti-inflammatory and anticancer agents through selectively targeting COX-2 | Shaker, Ahmed M M; Shahin, Mai I. ; AboulMagd, Asmaa M; Abdel Aleem, Seham A; Abdel-Rahman, Hamdy M; Abou El Ella, Dalal |
| 7 | 2022 | Novel Azine Linked Hybrids of 2-Indolinone and Thiazolodinone Scaffolds as CDK2 Inhibitors with Potential Anticancer Activity: In Silico Design, Synthesis, Biological, Molecular Dynamics and Binding Free Energy Studies | Qayed, Wesam S; Hassan, Mostafa A; El-Sayed, Wael ; Rogério A Silva, José; Aboul-Fadl, Tarek |
| 8 | 1-Feb-2024 | Novel indolinone-tethered benzothiophenes as anti-tubercular agents against MDR/XDR M. tuberculosis: Design, synthesis, biological evaluation and in vivo pharmacokinetic study | Eldehna, Wagdy M.; Mahmoud, Sally Tarek; Elshnawey, Esraa R.; Elsayed, Zainab M.; Majrashi, Taghreed A.; El-Ashrey, Mohamed K.; Rashed, Mahmoud; Hemeda, Loah R.; Shoun, Aly A.; Elkaeed, Eslam B.; El Hassab, Mahmoud A.; Abdel-Aziz, Marwa M.; Shahin, Mai I. |
| 9 | 1-Dec-2017 | Novel quinoline-3-carboxamides (Part 2): Design, optimization and synthesis of quinoline based scaffold as EGFR inhibitors with potent anticancer activity | Aly, Rasha M.; Serya, Rabah ; El-Motwally, Amira M.; Abbas, Safinaz; Abou El Ella, Dalal ; Esmat, Ahmed |
| 10 | Aug-2020 | Scaffold hopping and redesign approaches for quinazoline based urea derivatives as potent VEGFR-2 inhibitors | Hadi, Soha R Abd El; Soliman, Dalia H; Elrazaz, Eman ; Khaled A M Abouzid ; Lasheen, Deena S. |
| 11 | 29-Sep-2025 | Straightforward synthesis and in silico evaluation of pyrazolylthiazolidinone derivatives as prospective antiproliferative agents | Ramadan, Sayed ; Gomha, Sobhi M; El-Helw, Eman A. E. |
| 12 | Oct-2025 | Straightforward synthesis and in silico evaluation of pyrazolylthiazolidinone derivatives as prospective antiproliferative agents | Ramadan, Sayed K. ; Gomha, Sobhi M; Eman A. E. El-Helw |
| 13 | Feb-2022 | Structure-based design and synthesis of conformationally constrained derivatives of methyl-piperidinopyrazole (MPP) with estrogen receptor (ER) antagonist activity | Ragab, Mahmoud A; Elagawany, Mohamed; Daabees, Hoda; Ahmed, Al-Shaimaa F; Awad, Eman M; Billon, Cyrielle; Elgendy, Bahaa; Abouzid, Khaled ; Kassab, Shaymaa E |
| 14 | Jan-2020 | Synthesis and antimicrobial evaluation of new halogenated 1,3-Thiazolidin-4-ones | Hammad, Shaymaa G; El-Gazzar, Marwa G; Abutaleb, Nader S; Li, Daoyi; Ramming, Isabell; Shekhar, Aditya; Abdel-Halim, Mohammad; Elrazaz, Eman ; Seleem, Mohamed N; Bilitewski, Ursula; El-Hossary, Ebaa M; Khaled A M Abouzid |
| 15 | 2026 | Synthesis and biological evaluation of novel heterocyclic compounds derived from ammonium thiocyanate for control of Culex pipiens and Musca domestica. | Ghareeb, Eman A; Kamal, Mahmoud; Farag, Shaimaa M; Ammar, Asmaa M; Mahmoud, Naglaa FH; Eman A. E. El-Helw |
| 16 | 2025 | Synthesis of tetra-substituted thiophene derivatives as potential hits combating antibiotic resistant bacteria ESKAPE | AboulMagd, Asmaa M; Shaker, Ahmed MM; Farag, Paula S; aya ibrahim hassaballah ; Hemdan, Magdy M; Abd El-Mawgoud, Heba K |
| 17 | Jul-2021 | Synthesis, DFT, and eco-friendly insecticidal activity of some N-heterocycles derived from 4-((2-oxo-1,2-dihydroquinolin-3-yl)methylene)-2-phenyloxazol-5(4H)-one | Ghareeb, Eman A; Mahmoud, Naglaa F H; El-Bordany, Eman A; El-Helw, EAE |
| 18 | Sep-2021 | Synthesis, in vitro biological investigation, and molecular dynamics simulations of thiazolopyrimidine based compounds as corticotrophin releasing factor receptor-1 antagonists | Elgiushy, Hossam R; Abou-Taleb, Nageh A; Holz, George G; Chepurny, Oleg G; Pirmettis, Ioannis; Kakabakos, Sotirios; Karageorgos, Vlasios; Liapakis, George; Albohy, Amgad; Abouzid, Khaled ; Hammad, Sherif F |
| 19 | 27-Dec-2024 | Synthesis, in vivo evaluation, and in silico molecular docking of benzo[h]quinoline derivatives as potential Culex pipiens L. larvicides | Ramadan, Sayed ; Hosni, Eslam M; Kamal, Mahmoud ; El-Helw, Eman A. E. ; Hashem, Ahmed ; Wael Abou-Elmagd |
| 20 | 2024 | Synthesis, insecticidal Activity, and molecular docking analysis of some benzo[h]quinoline derivatives against Culex pipiens L. Larvae | Hosni, Eslam M.; Mahmoud Kamal ; Sayed Karam Ramadan Emam ; Eman A.E. El-Helw ; Hashem, Ahmed |
